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DOI 10.3109/14756366.2016.1170014

Медицинская библиотека · Journal of enzyme inhibition and medicinal chemistry · 2016

The synthesis of some β-lactams and investigation of their metal-chelating activity, carbonic anhydrase and acetylcholinesterase inhibition profiles.

Turan Burhanettin, Şendil Kivilcim, Şengül Emin, Gültekin Mehmet Serdar, Taslimi Parham, Gulçin İlhami, Supuran Claudiu T

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Аннотация

β-Lactam antibiotics are a broad class of antibiotics, consisting of all antibiotic agents that contain a β-lactam ring in their molecular structures. Synthesis of β-lactam analogs, which are containing dichloride atoms and N-methyl, N-aromatic rings, was achieved by Schiff bases and dichloroketene compounds. All the synthesized imines and β-lactam analogs were tested against two physiologically relevant carbonic anhydrase isozymes (hCA I and II) and acetylcholinesterase (AChE). They demponstrated effective inhibitory profiles with Ki values in ranging of 3.22-11.18 nM against hCA I, 3.74-10.41 nM against hCA II, and 0.50-1.57 nM against AChE. On the other hand, acetazolamide and dorzolamide clinically used as CA inhibitors, showed Ki value of 170.34 and 129.26 nM against hCA I, and 115.43 and 135.67 nM against hCA II, respectively. Also, tacrine used as standard AChE inhibitor showed Ki value of 5.70 nM against AChE.

Для цитирования: Turan Burhanettin, Şendil Kivilcim, Şengül Emin, Gültekin Mehmet Serdar, Taslimi Parham, Gulçin İlhami, Supuran Claudiu T. The synthesis of some β-lactams and investigation of their metal-chelating activity, carbonic anhydrase and acetylcholinesterase inhibition profiles.. Journal of enzyme inhibition and medicinal chemistry. 2016. DOI: 10.3109/14756366.2016.1170014.

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